Table 1 Suzuki–Miyaura cross-coupling of 15a and 16a^a

^aReaction conditions: 15a (47.0 mg, 0.1 mmol), 16a (27.6 mg, 0.2 mmol), catalyst (5 mol%), and base (3.0 equiv), in 1 mL solvent under nitrogen atmosphere for 12 h
^bIsolated yield
^cThe reaction was run at rt for 5 h
^dThe reaction was performed with 6.6 g of 15a and was quenched until 15a had disappeared as monitored by TLC

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