Table 1 Summary of the helicity and the macrocyclization yields of the stapled peptides.

Peptide	Fluoro substrates	Helicity (%)	Yield (%)	Peptide	Fluoro substrates	Helicity (%)	Yield (%)
29	l_N, _Cl	24	22	57	l_i, _i+4l	41	64
31	l_N, _Cl	21	23	58	l_i, _i+4d	39	61
33	l_N, _Cl	23	27	59	d_i, _i+4l	13	58
35	l_i, _i+4l	24	55	60	l_i, _i+4l	50	59
36	l_i, _i+4l	29	59	61	l_i, _i+4d	45	51
37	l_i, _i+4l	18	49	62	d_i, _i+4L	9	56
38	l_i, _i+4l	25	52	63^a	S₅, S₅	52	51
39	l_i, _i+4l	46	63	70	l_i, _i+4l	84	64
40	l_i, _i+4l	17	52	72	l_i, _i+4d	85	61
42	d_i, _i+4d	14	58	73^a	S₅, S₅	88	37
43	d_i, _i+4d	28	62	75	li, _i+4l	74	74
44	d_i, _i+4d	31	60	77	l_i, _i+4d	70	73
45	d_i, _i+4d	25	55	78^a	S₅, S₅	73	42
46	d_i, _i+4d	13	59	80	l_i, _i+7l	36	65
47	d_i, _i+4d	19	65	81	l_i, _i+7l	42	69
49	l_i, _i+4d	25	54	82	l_i, _i+7l	61	74
50	l_i, _i+4d	14	43	83	l_i, _i+7l	16	55
51	l_i, _i+4d	44	58	85	l_i, _i+7d	40	69
53	d_i, _i+4l	19	39	86	l_i, _i+7d	37	71
54	d_i, _i+4l	5	50	87	l_i, _i+7d	64	79
55	d_i, _i+4l	8	51	88	l_i, _i+7d	18	55
56^a	S₅, S₅	48	73	89^a	R₈, S₅	65	58

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