Fig. 3: Scope of para-arylation.
From: Expanding chemical space by para-C−H arylation of arenes
a Scope of the reaction with O-glycosylated aryl iodides. b Scope of para-C–H arylation with iodo-containing drugs. Reaction conditions: arene (1 equiv.), (hetero)aryl iodide (1 equiv.), Pd(OAc)2 (10 mol%), N-Fmoc-Gly-OH (20 mol%), Ag2SO4 (2 equiv.), Cr2Cu2O5 (2 equiv.), LiOAc.2H2O (0.5 equiv.), HFIP, 80 °C, 24 h. # the isomer for 5uk was not separated clearly.
