Fig. 5: Gram-scale experiment and synthetic application.

a Gram-scale experiment. b One-pot asymmetric hydroamidation w/o isolation of alkenyl boronate. c Concise synthetic route to Vaborbactam.
a Gram-scale experiment. b One-pot asymmetric hydroamidation w/o isolation of alkenyl boronate. c Concise synthetic route to Vaborbactam.