Table 2 Kinetic parameters of MaAT8824 for compounds 1, 3, 5 and 6
Substrate | Acyl donor | Acylation site | Km [μM] | kcat [s−1] | kcat/Km [s−1 M−1] |
---|---|---|---|---|---|
1 | Acetyl-CoA | 12-OH | 64.1 | 0.020 | 318.43 |
3 | Acetyl-CoA | 12-OH | 205.1 | 0.037 | 180.2 |
5 | Acetyl-CoA | 12-OH | 390.7 | 0.014 | 35.1 |
6 | Acetyl-CoA | 3-OH | 232.5 | 0.024 | 106.8 |