Table 2 Scope for benzazaborines from acyclic ketones and drug moleculesa

From: Organocatalysed three-component modular synthesis of BN isosteres and BN-2,1-azaboranaphthalenes via Wolff-type rearrangement

  1. aIsolated yields are mentioned.
  2. bReaction was carried out with 300 mol% pyrrolidine.
  3. cReaction was carried out with at 4.4 mmol scale, 72% yield (0.80 g).