Table 1 IC50 values and 95% confidence interval (in nM) of the competitive binding assay on INS-1 cells.
From: Preclinical evaluation of PAC1 targeting with radiolabeled Maxadilan
Peptide | IC50 (nM) | 95% confidence interval (nM) |
|---|---|---|
Maxadilan | 3.2 | 2.1–4.9 |
Maxadilan-DTPA | 13.2 | 8.8–19.8 |
DTPA-Maxadilan | 18.3 | 13.2–25.3 |
Maxadilan-DTPA- NatIn | 21.0 | 13.7–32.2 |
NatIn-DTPA-Maxadilan | 21.0 | 11.8–37.3 |