Table 1 Pharmacokinetic parameters of empagliflozin (EG) following oral administration of one JARDIANCE tablet nominally containing 25 mg of EG.
Pharmacokinetic parameters | Empagliflozin |
---|---|
Cmax (nMol/L), Mean ± S.D. (% C.V.) | 576 ± 86 (14.93) |
Tmax (hours), Median (range) | 1.5, (1–2) |
t 1/2 (hours), Mean ± S.D. (% C.V.) | 6.1 ± 1.2 (19.67) |
Elimination rate constant (h−1), Mean ± S.D. (% C.V.) | 0.10012 ± 0.02156 (19.25) |
AUC0−t (12) (nMol.h/L), Mean ± S.D. (% C.V.) | 2806 ± 234 (8.34) |
AUC0-inf (nMol.h/L), Mean ± S.D. (% C.V.) | 4103 ± 427 (10.41) |