Table 2 Effect of dinapinones on neutral lipid synthesis in CHO-K1 cells.
Compound | IC50 (μM) | |
---|---|---|
TG | CE | |
DPA1 | >12 | >12 |
DPA2 | 0.65 | >12 |
DPAmix | 0.054 | 0.18 |
DPAB1 | >12 | >12 |
DPAB2 | 1.1 | >12 |
DPABmix | 0.030 | 0.089 |
DPAC1 | >11 | >11 |
DPAC2 | >11 | >11 |
DPACmix | >11 | >11 |
DPAD1 | >12 | >12 |
DPAD2 | 4.2 | >12 |
DPADmix | 0.20 | 4.4 |
DPAE1 | 4.8 | >11 |
DPAE2 | 4.3 | >11 |
DPAEmix | 0.13 | 6.3 |