Fig. 5: Anhydrotetracycline and analogues inhibit enzymatic inactivation of latest-generation tetracyclines by Tet(X7). | Communications Biology

Fig. 5: Anhydrotetracycline and analogues inhibit enzymatic inactivation of latest-generation tetracyclines by Tet(X7).

From: Tetracycline-inactivating enzymes from environmental, human commensal, and pathogenic bacteria cause broad-spectrum tetracycline resistance

Fig. 5

a In vitro, anhydrotetracycline, anhydrochlortetracycline, and anhydrodemeclocycline inhibit Tet(X) modification of tigecycline. Likewise, anhydrotetracycline and anhydrodemeclocycline inhibit in vitro enzymatic modification of tigecycline (b), eravacycline (c), and omadacycline (d) by Tet(X7). Error bars represent standard deviation for three independent trials.

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