Table 3 Enzymatic activities and IC50 values of BCArg mutant and 2b-modified BCArg mutant.
From: N-Terminal selective modification of peptides and proteins using 2-ethynylbenzaldehydes
Sample | BCArg mutant | 2b-modified BCArg mutant |
---|---|---|
Specific activity (U/mg) | 443.96 ± 27.50 | 313.68 ± 4.01 |
IC50 values for MDA-MB-231 (U/mL) | 4.608 ± 0.995 | 5.491 ± 1.564 |
IC50 values for MDA-MB-468 (U/mL) | 4.772 ± 1.137 | 5.631 ± 2.410 |