Table 1 Kidney cells and mutation status in GDSC database

From: PI3Kβ Inhibitor TGX221 Selectively Inhibits Renal Cell Carcinoma Cells with Both VHL and SETD2 mutations and Links Multiple Pathways

Cell line

COSMIC

Cell type

Mutation

IC50 (Log10)

VHL

SETD2

BAP1

PBRM1

NOTCH1

769-P

910922

Clear cell renal cell carcinoma

*

 

*

   

786-0

905947

Clear cell renal cell carcinoma

*

     

A498

905948

Clear cell renal cell carcinoma

*

*

   

−1.085304

A704

905948

Renal cell adenocarcinoma

*

*

    

ACHN

905950

Clear cell renal cell carcinoma

   

*

  

BB65-RCC

753533

Renal cell adenocarcinoma

*

    

4.721833

BFTC-909

910698

Transitional cell carcinoma

   

*

  

CAKI-1

905963

Clear cell renal cell carcinoma

 

*

    

CAL-54

910952

Renal cell carcinoma

      

G-401

907299

Renal rhabdoid tumour

      

LB1047-RCC

753577

Renal cell carcinoma

   

*

 

4.183081

LB2241-RCC

753578

Renal cell carcinoma

     

4.125849

LB996-RCC

753585

Renal cell carcinoma

 

*

   

2.589532

OS-RC-2

909250

Clear cell renal cell carcinoma

*

  

*

 

0.800791

RCC10RGB

909974

Renal cell carcinoma

*

 

*

  

2.415331

RXF393

905978

Hypernephroma

     

1.904166

SK-NEP-1

909730

Wilm's Tumour

     

4.933583

SN12C

905979

Renal cell carcinoma

  

*

   

TK10

905980

Renal cell carcinoma

     

4.287613

U031

905981

Renal cell carcinoma

      

VMRC-RCZ

909781

Renal cell carcinoma

*