Table 1 Binding affinities and selectivity of complex 1 for various oligonucleotides, determined by the FID assay.
DC50a (μM) | Selectivity against ds26b | |
---|---|---|
HTelo | 1.01 (0.03) | 9.81 |
KRAS m(1:5:1) | 2.28 (0.10) | 4.34 |
KRAS m(1:9:1) | 2.35 (0.09) | 4.22 |
c-Kit | 3.58 (0.28) | 2.77 |
c-Myc | 7.15 (0.17) | 1.39 |
ds26 | 9.91 (0.55) | — |
HIF1α | 10.20 (0.54) | 0.97 |
hTERT | 10.51 (0.61) | 0.94 |
VEGF | 11.58 (0.41) | 0.86 |