Table 6 Absorption properties of oleocanthal, oleacein, luteolin, tyrosol, ezetimibe, and bempedoic acid.
Absorbsion properties | Oleocanthal | Oleacein | Luteolin | Tyrosol | Ezetimibe | Bempedoic acid |
---|---|---|---|---|---|---|
Caco-2 Permeability | -4.789 | -4.865 | -5.192 | -4.856 | -5.019 | -5.154 |
MDCK Permeability | -4.691 | -4.659 | -4.799 | -4.689 | -4.722 | -4.764 |
PAMPA | 0.753 | 0.723 | 0.345 | 0.773 | 0.042 | 0.999 |
Pgp-inhibitor | 0.205 | 0.04 | 0.001 | 0.018 | 0.974 | 0.0 |
Pgp-Substrate | 0.768 | 0.329 | 0.209 | 0.775 | 0.031 | 0.297 |
HIA | 0.01 | 0.097 | 0.015 | 0.093 | 0.0 | 0.898 |
F20% | 0.691 | 0.987 | 0.925 | 0.226 | 0.007 | 0.231 |
F30% | 0.697 | 0.99 | 0.992 | 0.183 | 0.073 | 0.281 |
F50% | 0.998 | 1 | 0.998 | 0.975 | 0.007 | 0.441 |