Table 8 Metabolic properties of oleocanthal, oleacein, luteolin, tyrosol, ezetimibe, and bempedoic acid.
Metablosim properties | Oleocanthal | Oleacein | Luteolin | Tyrosol | Ezetimibe | Bempedoic acid |
---|---|---|---|---|---|---|
CYP1A2 inhibitor | 0.007 | 0.003 | 1.0 | 0.023 | 0.003 | 0.0 |
CYP2C19 inhibitor | 0.498 | 0.372 | 0.01 | 0.013 | 0.017 | 0.0 |
CYP2C9 inhibitor | 0.972 | 0.139 | 0.001 | 0.016 | 0.321 | 0.015 |
CYP2D6 inhibitor | 0.005 | 0.001 | 0.578 | 0.02 | 0.64 | 0.0 |
CYP3A4 inhibitor | 0.999 | 0.999 | 0.998 | 0.036 | 0.006 | 0.001 |