Table 1 Michaelis–Menten kinetics of MERTK at different BMS794833 concentrations.

From: BMS794833 inhibits macrophage efferocytosis by directly binding to MERTK and inhibiting its activity

BMS794833

0 nM

10 nM

20 nM

30 nM

40 nM

50 nM

Vmax

20,805 ± 488

20,871 ± 176

20,242 ± 178

20,948 ± 265

21,462 ± 141

21,639 ± 361

Km (ÎĽM)

23.52 ± 0.54

26.88 ± 0.63

36.98 ± 1.30

54.52 ± 0.30

65.86 ± 0.82

79.45 + 3.21

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