Table 1 Inhibition of [3H]-l-leucine transport into HT-29 cells by JX-075, JX-078, and JX-119.
From: Mechanism of substrate transport and inhibition of the human LAT1-4F2hc amino acid transporter
Compound | IC50 [nM] | 95% Confidence interval [nM] |
|---|---|---|
JX-075 | 165 | 151–180 |
JX-078 | 121 | 108–137 |
JX-119 | 234 | 87–293 |