Fig. 1: Direct deaminative functionalization of aromatic amines. | Nature

Fig. 1: Direct deaminative functionalization of aromatic amines.

From: Direct deaminative functionalization with N-nitroamines

Fig. 1: Direct deaminative functionalization of aromatic amines.

a, Relative commercial availability of common aryl donors used in cross-coupling reactions (data retrieved from the Reaxys database). b, Recent advances in deaminative functionalization of aromatic amines10,11,14. c, Aromatic amines as direct precursors to aryl donors with in situ rapid diversification (this work). Het., heterocycle.

Back to article page