Table 2 Biodistribution data of 188Re-labeled peptides following intravenous injection into A549 tumor-bearing nude mice.
Organs | Uptake (%ID/g) | Tumor-organ ratio | ||||||
|---|---|---|---|---|---|---|---|---|
QKRKRKKSRKKH | RKRKRKKSRYIVLS | QKRKRKKSRKKH | RKRKRKKSRYIVLS | |||||
2 h | 6 h | 2 h | 6 h | 2 h | 6 h | 2 h | 6 h | |
blood | 10.9 ± 1.72 | 10.9 ± 1.72 | 6.97 ± 1.36 | 3.26 ± 0.33 | 0.29 | 0.78 | 1.91 | 1.33 |
heart | 5.5 ± 2.35 | 5.5 ± 2.35 | 2.31 ± 0.44 | 1.61 ± 0.3 | 0.58 | 1.09 | 5.76 | 2.70 |
liver | 11.88 ± 2.92 | 11.88 ± 2.92 | 14.46 ± 3.38 | 12.85 ± 1.05 | 0.27 | 0.44 | 0.92 | 0.34 |
spleen | 2.41 ± 0.7 | 2.41 ± 0.7 | 8.73 ± 0.8 | 4.41 ± 2 | 1.33 | 1.43 | 1.52 | 0.99 |
lung | 2.93 ± 1.31 | 2.93 ± 1.31 | 1.69 ± 0.51 | 0.91 ± 0.57 | 1.09 | 2.32 | 7.88 | 4.78 |
kidney | 33.79 ± 3.39 | 33.79 ± 3.39 | 48.33 ± 3.89 | 22.81 ± 4.84 | 0.09 | 0.14 | 0.28 | 0.19 |
stomach | 6.02 ± 2.83 | 6.02 ± 2.83 | 4.18 ± 0.8 | 7.44 ± 1.94 | 0.53 | 0.71 | 3.18 | 0.58 |
bone | 3.36 ± 2.09 | 3.36 ± 2.09 | 2.25 ± 0.75 | 3.45 ± 1.5 | 0.95 | 3.32 | 5.92 | 1.26 |
muscle | 0.71 ± 0.34 | 0.71 ± 0.34 | 2.49 ± 0.7 | 0.79 ± 0.1 | 4.51 | 4.35 | 5.35 | 5.51 |
brain | 0.61 ± 0.22 | 0.61 ± 0.22 | 0.34 ± 0.13 | 0.38 ± 0.15 | 5.25 | 7.96 | 39.15 | 11.45 |
tumor | 3.2 ± 1.16 | 3.2 ± 1.16 | 13.31 ± 1.17 | 4.35 ± 0.85 | — | — | — | — |