Table 1 Main characteristics of the patients at day of inclusion.

From: Impact of UGT1A1 polymorphisms on Raltegravir and its glucuronide plasma concentrations in a cohort of HIV-1 infected patients

Number of patients included

96

Age, years (mean ± SD)

52.6 ± 11.7

Body Mass Index, kg/m2 (mean ± SD)

25.8 ± 4.4

Gender, n (%) male

56 (58%)

Ethnic origin, n (%)

    Caucasian

59 (61%)

    African

34 (35%)

    Asian

2

    South American

1

Co-administered ARV drugs

NRTI

ABC/3TC (n = 8), FTC/TDF (=38), 3TC (n = 17), TDF245mg (n = 8), ABC 600 (n = 1), NRTI-free (n = 25)

NNRTI

ETR (n = 17), NVP (n = 3), EFV/FTC/TDF (n = 2)

PI

DRV (n = 39), ATV (n = 3), LPV/r (n = 3)

MVC

n = 13

CD4 cell count, cells per μl (median [min-max])

620 [88–1418]

Nadir CD4 cell count, cells per μl (median [min-max])

119 [2–402]

HIV-1 RNA < 40 copies per mL, n (%)

90 (94%)

HIV-1 RNA > 40 copies per mL, n (%)

copies per mL (median [min-max])

6 (6%)

69 [41–152]

Duration of treatment, months (mean ± SD)

42.1 ± 23.7

Post-intake delay, hours (mean [CI95%])

15 [14.2–15.8]

  1. ARV: antiretroviral, NNRTI: Non-Nucleoside Reverse Transcriptase Inhibitor, NRTI: Nucleoside Reverse Transcriptase Inhibitor, PI: protease inhibitor, DRV: darunavir, ATV: atazanavir, LPV/r: Lopinavir/ritonavir, MVC: maraviroc ETR: etravirine, NVP: nevirapine, ABC: abacavir, 3TC: lamivudine, FTC: emtricitabine, TDF: tenofovir disoproxil fumarate, NRTI-free: without any NRTI.