Figure 2

Per amino-acid interaction energy map for a dataset of hydroxy aryl aldehyde (HAA) class of IRE1 endoribonuclease inhibitors docked inside the binding site of MKC9989 using conventional docking studies (PDB code: 4PL3). (A) Electrostatic energy values (kcal mol−1); (B) Hydrophobic score (arbitrary units).