Table 1 Ki values (expressed in µM, mean ± SD, n = 6) of the ortho-, meta- and para- substituted compounds, FET and l-phenylalanine.
From: New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma
Compound | Ki value (µM) | Compound | Ki value (µM) |
|---|---|---|---|
| 16.09 ± 3.74 |
| 359.40 ± 47.10 |
| 48.95 ± 4.92 |
| 83.75 ± 28.10 |
| 85.55 ± 4.40 |
| >2000 |
| 307.20 ± 4.29 |
| 51.53 ± 7.80 |