Table 1 Associated constants of m-gate.

From: Characterization of a novel LQT3 variant with a selective efficacy of mexiletine treatment

 

\({{\boldsymbol{V}}}_{{\bf{h}}(m{\boldsymbol{\infty }})}\)

k m

\({{\boldsymbol{V}}}_{{{\bf{h}}}_{{{\boldsymbol{m}}}_{{\boldsymbol{\tau }}}}}\)

a m

b m

c m

d m

WT

−36.445

−4.519

−52.000

1.206

−46.861

−126.579

0.226

A1656D

−44.694

−5.369

−68.764

5.078

196.176

85.086

0

Mexiletine

−47.173

−4.998

−62.604

6.202

256.571

126.690

0.106

Flecainide

−54.609

−3.615

−61.536

1.347

122.632

53.127

0.394

Ranolazine

−50.270

−4.950

−63.290

3.394

161.294

90.427

0.135