Table 3 Summary of in vitro properties and in vitro and in vivo stability of [18F]21 (see also Supplementary Fig. S5).
logD7.4 | Plasma protein binding | Stability in human serum and plasma (in vitro, after 60 min) | Stability in mouse blood (in vivo, 10 min p.i.) |
|---|---|---|---|
− 3.1 ± 0.1 (n = 3) | 10% | 99% | 30% |