Table 2 Biodistribution of the 64+67Cu-ODDA complex in tumor-bearing mice at various time points.
Organ/tissue | 0.5 h p.i | 1 h p.i | 2 h p.i | 4 h p.i | 12 h p.i | 24 h p.i |
|---|---|---|---|---|---|---|
Tumor (Right Thigh) | 7.8 ± 0.4 | 13.5 ± 1.1 | 18.0 ± 0.3 | 7.8 ± 0.7 | 4.5 ± 0.4 | 2.1 ± 0.2 |
Left Muscle (Control Thigh) | 1.4 ± 0.2 | 2.2 ± 0.3 | 1.9 ± 0.2 | 0.9 ± 0.2 | 0.6 ± 0.3 | 0.3 ± 0.1 |
Liver | 6.0 ± 0.7 | 5.5 ± 0.6 | 4.8 ± 0.5 | 3.9 ± 0.4 | 2.8 ± 0.3 | 1.9 ± 0.2 |
Kidneys | 10.5 ± 0.8 | 11.2 ± 0.7 | 10.8 ± 0.6 | 9.6 ± 0.5 | 7.4 ± 0.4 | 5.1 ± 0.3 |
Lungs | 5.8 ± 0.5 | 4.9 ± 0.4 | 4.0 ± 0.4 | 3.1 ± 0.3 | 2.2 ± 0.2 | 1.5 ± 0.2 |
Spleen | 2.4 ± 0.3 | 2.2 ± 0.3 | 2.0 ± 0.2 | 1.7 ± 0.2 | 1.2 ± 0.2 | 0.8 ± 0.1 |
Heart | 2.0 ± 0.3 | 1.8 ± 0.3 | 1.6 ± 0.2 | 1.3 ± 0.2 | 1.0 ± 0.2 | 0.6 ± 0.1 |
Bone | 2.5 ± 0.3 | 2.3 ± 0.2 | 2.0 ± 0.2 | 1.6 ± 0.2 | 1.3 ± 0.2 | 1.0 ± 0.2 |
Intestine | 2.8 ± 0.4 | 2.5 ± 0.3 | 2.2 ± 0.3 | 1.9 ± 0.2 | 1.4 ± 0.2 | 0.9 ± 0.1 |
Blood | 4.0 ± 0.5 | 3.5 ± 0.4 | 3.0 ± 0.3 | 2.4 ± 0.3 | 1.8 ± 0.2 | 1.0 ± 0.2 |
T/NT | 5.6 | 6.1 | 9.4 | 8.6 | 7.5 | 7.0 |
Tumor/Blood | 1.9 | 3.9 | 6.0 | 3.3 | 2.5 | 2.1 |