Table 1 Encapsulation efficiency (EE) and drug loading efficiency (DLE) of the liposomes.
Liposome | DOPC (mg/mL) | Cholesterol (mg/mL) | DSPE(PEG)2000-OMe (mg/mL) | TTP (mg/mL) | E (mg/mL) | G (mg/mL) | DLE (%) | EE (%) |
|---|---|---|---|---|---|---|---|---|
L | 3.93 | 0.965 | 0.140 | 0.452 | – | – | – | – |
E-L | 3.93 | 0.965 | 0.140 | 0.452 | 0.4 | – | 7.29 | 100 |
G-L | 3.93 | 0.965 | 0.140 | 0.452 | – | 0.120 | 2.2 | 30 |
EG-L | 3.93 | 0.965 | 0.140 | 0.452 | 0.4 | 0.120 | 7.29 (E), 2.2 (G) | 100 (E), 30 (G) |