Cell‐Active, Irreversible Covalent Inhibitors Targeting a Surface‐Exposed Non‐Catalytic Lysine on Aurora a Kinase by Using Squarate Chemistry

Journal:
Angewandte Chemie International Edition
Published:
Affiliations:
4
Authors:
13
Institutions Authors Share
State Key Laboratory of Bioactive Molecules and Druggability Assessment, JNU, China
9.000000
0.69
National University of Singapore (NUS), Singapore
3.000000
0.23
Guangdong Second Provincial General Hospital, China
0.500000
0.04
Jinan University (JNU), China
0.500000
0.04