Scalable Synthesis of a Dual TLR7/8 Agonist via Highly Selective N2-Alkylation of 1H-Pyrazolo[4,3-d]pyrimidine

Journal:
Organic Letters
Published:
DOI:
10.1021/acs.orglett.5c04092
Affiliations:
3
Authors:
7
Institutions Authors Share
Merck & Co, United States of America (USA)
4.000000
0.57
WuXi AppTec, China
3.000000
0.43