Asymmetric Synthesis of KRAS G12C Inhibitor MK-1084 via a Crystallization-Induced Diastereomer Transformation (CIDT)

Journal:
Organic Letters
Published:
DOI:
10.1021/acs.orglett.5c04646
Affiliations:
5
Authors:
25
Institutions Authors Share
Merck - Rahway, United States of America (USA)
19.000000
19.000000
0.76
Pharmaron, China
3.000000
0.12
Shanghai Syn-The-All Pharmaceutical Co. Ltd., China
3.000000
0.12