Modulating the Binding Kinetics of Bruton’s Tyrosine Kinase Inhibitors through Transition-State Effects

Journal:
Journal of the American Chemical Society
Published:
Affiliations:
7
Authors:
14
Institutions Authors Share
State University of New York at Stony Brook (SUNY Stony Brook), United States of America (USA)
8.166667
0.58
Enzymlogic, Spain
3.000000
0.21
Iowa State University, United States of America (USA)
2.000000
0.14
Cancer Research UK Cambridge Institute (CRUK-CI), University of Cambridge, United Kingdom (UK)
0.500000
0.04
University of Rochester Medical Center (URMC), UR, United States of America (USA)
0.333333
0.02